1. J. Li*, Y. Yao*, S. Zhang*, W. Wang, W. Bi, J. Lv, W. Hou#, P. Ma#, H. Xu#, Splint RNA-mediated Single-stranded DNA-Encoded Library Construction and Label-free Live Cell Selection, Chem. 2026, 12, 102945.
2. W. Zhou*, Y. Wang*, S. Zhang*, C. Zhang*, J. Pang, S. Hou, J. Li, Y. Yao, A. Su#, P. Ma#, H. Xu#, W. Hou#, Highly Selective and AI-Predictable Se-N Exchange Chemistry Between Benzoselenazolones and Boronic Acids for Programmable, Parallel, and DNA-Encoded Library Synthesis, Chem. Sci. 2026, 17, 225-239.
3. W. Hou*,#, X. Zhou*, Z. Yang*, H. Xia*, Y. Wang, K. Xu, S. Hou, S. Zhang, D. Cui, P. Ma, W. Zhou#, H. Xu#, Multicomponent Reaction Integrating Selenium(II)-Nitrogen Exchange (SeNEx) Chemistry and Copper-Catalyzed Azide-Alkyne Cycloaddition (CuAAC), Angew. Chem. Int. Ed. 2025, 64, e202500942.
4. W. Hou*, S. Zhang*, W. Yi#, P. Ma#, H. Xu#, DNA-Compatible Chemistry for DNA-Encoded Libraries and Beyond, Trends Chem. 2025, 7, 771-786.
5. H. Li*, Y. Liu*, S. Zhang*, L. Ma, Z. Zeng, Z. Zhou, V. Gandon, H. Xu#, W. Yi#, S. Wang#, Access to N-α-deuterated amino acids and DNA conjugates via Ca(II)-HFIP-mediated reductive deutero-amination of α-oxo-carbonyl compounds, Nat. Commun. 2025, 16, 1816.
6. W. Hou*,#, Y. Zhang*, F. Huang*, W. Chen*, Y. Gu, Y. Wang, J. Pang, H. Dong, K. Pan, S. Zhang, P. Ma, H. Xu#, Bioinspired Selenium‐Nitrogen Exchange (SeNEx) Click Chemistry Suitable for Nanomole‐Scale Medicinal Chemistry and Bioconjugation, Angew. Chem. Int. Ed. 2024, 63, e202318534.
7. P. Ma*, S. Zhang*, Q. Huang, Y. Gu, Z. Zhou, W. Hou#, W. Yi#, H. Xu#, Evolution of chemistry and selection technology for DNA-encoded library, Acta Pharm. Sin. B. 2024, 14, 492–516.
8. S. Zhang*, H. Zhang*, X. Liu*, P. Qi, T. Tan, S. Wang, H. Gao, H. Xu#, Z. Zhou#, W. Yi#, Mask and Release Strategy‐Enabled Diversity‐Oriented Synthesis for DNA‐Encoded Library, Adv. Sci. 2024, 11, 2307049.
9. Z. Zhou*, Y. Gu*, L. Wu*, Y. Wang*, H. Xu, L. Ma, Z. Zhang, J. Zhao, W. Zhang, W. Peng, G. Yang, X. Yu, H. Xu#, W. Yi#, Organo-Se BTSAs-enabled performance: From racemic and asymmetric synthesis to click chemistry application, Chem. 2023, 9, 3335–3346.
10. H. Xu*,#, Y. Wang*, H. Dong, Y. Zhang, Y. Gu, S. Zhang, Y. Meng, J. Li, X. Shi, Q. Ji, L. Liu, P. Ma, F. Ma#, G. Yang#, W. Hou#, Selenylation Chemistry Suitable for on‐Plate Parallel and On‐DNA Library Synthesis Enabling High‐Throughput Medicinal Chemistry, Angew. Chem. Int. Ed. 2022, 61, e202206516.
11. H. Xu*,#, T. Tan*, Y. Zhang, Y. Wang, K. Pan, Y. Yao, S. Zhang, Y. Gu, W. Chen, J. Li, H. Dong, Y. Meng, P. Ma#, W. Hou#, G. Yang#, Metal-Free and Open-Air Arylation Reactions of Diaryliodonium Salts for DNA-Encoded Library Synthesis, Adv. Sci. 2022, 9, 2202790.
12. S. Wang*, X. Shi*, J. Li*, Q. Huang, Q. Ji, Y. Yao, T. Wang, L. Liu, M. Ye, Y. Deng, P. Ma#, H. Xu#, G. Yang#, A Small Molecule Selected from a DNA‐Encoded Library of Natural Products That Binds to TNF‐α and Attenuates Inflammation In Vivo, Adv. Sci. 2022, 9, 2201258.
13. F. Ma, J. Li, S. Zhang, Y. Gu, T. Tan, W. Chen, S. Wang, H. Xu#, G. Yang#, R.A. Lerner#, Metal-Catalyzed One-Pot On-DNA Syntheses of Diarylmethane and Thioether Derivatives, ACS Catal. 2022, 12, 1639–1649.
14. W. Hou#, H. Xu#, Incorporating Selenium into Heterocycles and Natural Products─From Chemical Properties to Pharmacological Activities, J. Med. Chem. 2022, 65, 4436–4456.
15. W. Hou#, H. Dong, X. Zhang#, Y. Wang, L. Su, H. Xu#, Selenium as an Emerging Versatile Player in Heterocycles and Natural Products Modification, Drug Discov. Today, 2022, 27, 2268-2277
16. H. Gao*, S. Lin*, S. Zhang*, W. Chen, X. Liu, G. Yang, R.A. Lerner, H. Xu#, Z. Zhou#, W. Yi#, gem‐Difluoromethylene Alkyne‐Enabled Diverse C−H Functionalization and Application to the on‐DNA Synthesis of Difluorinated Isocoumarins, Angew. Chem. Int. Ed. 2021, 60, 1959–1966.
17. Q. Zheng*, H. Xu*, H. Wang, W.H. Du, N. Wang, H. Xiong, Y. Gu, L. Noodleman, K.B. Sharpless#, G. Yang#, P. Wu#, Sulfur [18F]Fluoride Exchange Click Chemistry Enabled Ultrafast Late-Stage Radiosynthesis, J. Am. Chem. Soc. 2021, 143, 3753–3763.
18. H. Xu*, Y. Gu*, S. Zhang, H. Xiong, F. Ma, F. Lu, Q. Ji, L. Liu, P. Ma, W. Hou#, G. Yang#, R.A. Lerner#, A Chemistry for Incorporation of Selenium into DNA‐Encoded Libraries, Angew. Chem. Int. Ed. 2020, 59, 13273–13280.
19. H. Xu*, F. Ma*, N. Wang, W. Hou, H. Xiong, F. Lu, J. Li, S. Wang, P. Ma, G. Yang#, R.A. Lerner#, DNA‐Encoded Libraries: Aryl Fluorosulfonates as Versatile Electrophiles Enabling Facile On‐DNA Suzuki, Sonogashira, and Buchwald Reactions, Adv. Sci. 2019, 6, 1901551.
20. P. Ma*, H. Xu*, J. Li*, F. Lu, F. Ma, S. Wang, H. Xiong, W. Wang, D. Buratto, F. Zonta, N. Wang, K. Liu, T. Hua, Z. Liu, G. Yang#, R.A. Lerner#, Functionality independent DNA encoding of complex natural products, Angew. Chem. Int. Ed. 2019, 58, 9254-9261.