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代表性论文:*第一作者,#通讯作者)

1. J. Li*, Y. Yao*, S. Zhang*, W. Wang, W. Bi, J. Lv, W. Hou#, P. Ma#, H. Xu#, Splint RNA-mediated Single-stranded DNA-Encoded Library Construction and Label-free Live Cell Selection, Chem. 2026, 12, 102945.

2. W. Zhou*, Y. Wang*, S. Zhang*, C. Zhang*, J. Pang, S. Hou, J. Li, Y. Yao, A. Su#, P. Ma#, H. Xu#, W. Hou#, Highly Selective and AI-Predictable Se-N Exchange Chemistry Between Benzoselenazolones and Boronic Acids for Programmable, Parallel, and DNA-Encoded Library Synthesis, Chem. Sci. 2026, 17, 225-239.

3. W. Hou*,#, X. Zhou*, Z. Yang*, H. Xia*, Y. Wang, K. Xu, S. Hou, S. Zhang, D. Cui, P. Ma, W. Zhou#, H. Xu#, Multicomponent Reaction Integrating Selenium(II)-Nitrogen Exchange (SeNEx) Chemistry and Copper-Catalyzed Azide-Alkyne Cycloaddition (CuAAC), Angew. Chem. Int. Ed. 2025, 64, e202500942.

4. W. Hou*, S. Zhang*, W. Yi#, P. Ma#, H. Xu#, DNA-Compatible Chemistry for DNA-Encoded Libraries and Beyond, Trends Chem. 2025, 7, 771-786.

5. H. Li*, Y. Liu*, S. Zhang*, L. Ma, Z. Zeng, Z. Zhou, V. Gandon, H. Xu#, W. Yi#, S. Wang#, Access to N-α-deuterated amino acids and DNA conjugates via Ca(II)-HFIP-mediated reductive deutero-amination of α-oxo-carbonyl compounds, Nat. Commun. 2025, 16, 1816.

6. W. Hou*,#, Y. Zhang*, F. Huang*, W. Chen*, Y. Gu, Y. Wang, J. Pang, H. Dong, K. Pan, S. Zhang, P. Ma, H. Xu#, Bioinspired SeleniumNitrogen Exchange (SeNEx) Click Chemistry Suitable for NanomoleScale Medicinal Chemistry and Bioconjugation, Angew. Chem. Int. Ed. 2024, 63, e202318534.

7. P. Ma*, S. Zhang*, Q. Huang, Y. Gu, Z. Zhou, W. Hou#, W. Yi#, H. Xu#, Evolution of chemistry and selection technology for DNA-encoded library, Acta Pharm. Sin. B. 2024, 14, 492–516.

8. S. Zhang*, H. Zhang*, X. Liu*, P. Qi, T. Tan, S. Wang, H. Gao, H. Xu#, Z. Zhou#, W. Yi#, Mask and Release StrategyEnabled DiversityOriented Synthesis for DNAEncoded Library, Adv. Sci. 2024, 11, 2307049.

9. Z. Zhou*, Y. Gu*, L. Wu*, Y. Wang*, H. Xu, L. Ma, Z. Zhang, J. Zhao, W. Zhang, W. Peng, G. Yang, X. Yu, H. Xu#, W. Yi#, Organo-Se BTSAs-enabled performance: From racemic and asymmetric synthesis to click chemistry application, Chem. 2023, 9, 3335–3346.

10. H. Xu*,#, Y. Wang*, H. Dong, Y. Zhang, Y. Gu, S. Zhang, Y. Meng, J. Li, X. Shi, Q. Ji, L. Liu, P. Ma, F. Ma#, G. Yang#, W. Hou#, Selenylation Chemistry Suitable for onPlate Parallel and OnDNA Library Synthesis Enabling HighThroughput Medicinal Chemistry, Angew. Chem. Int. Ed. 2022, 61, e202206516.

11. H. Xu*,#, T. Tan*, Y. Zhang, Y. Wang, K. Pan, Y. Yao, S. Zhang, Y. Gu, W. Chen, J. Li, H. Dong, Y. Meng, P. Ma#, W. Hou#, G. Yang#, Metal-Free and Open-Air Arylation Reactions of Diaryliodonium Salts for DNA-Encoded Library Synthesis, Adv. Sci. 2022, 9, 2202790.

12. S. Wang*, X. Shi*, J. Li*, Q. Huang, Q. Ji, Y. Yao, T. Wang, L. Liu, M. Ye, Y. Deng, P. Ma#, H. Xu#, G. Yang#, A Small Molecule Selected from a DNAEncoded Library of Natural Products That Binds to TNFα and Attenuates Inflammation In Vivo, Adv. Sci. 2022, 9, 2201258.

13. F. Ma, J. Li, S. Zhang, Y. Gu, T. Tan, W. Chen, S. Wang, H. Xu#, G. Yang#, R.A. Lerner#, Metal-Catalyzed One-Pot On-DNA Syntheses of Diarylmethane and Thioether Derivatives, ACS Catal. 2022, 12, 1639–1649.

14. W. Hou#, H. Xu#, Incorporating Selenium into Heterocycles and Natural Products─From Chemical Properties to Pharmacological Activities, J. Med. Chem. 2022, 65, 4436–4456.

15. W. Hou#, H. Dong, X. Zhang#, Y. Wang, L. Su, H. Xu#, Selenium as an Emerging Versatile Player in Heterocycles and Natural Products Modification, Drug Discov. Today, 2022, 27, 2268-2277

16. H. Gao*, S. Lin*, S. Zhang*, W. Chen, X. Liu, G. Yang, R.A. Lerner, H. Xu#, Z. Zhou#, W. Yi#, gemDifluoromethylene AlkyneEnabled Diverse C−H Functionalization and Application to the onDNA Synthesis of Difluorinated Isocoumarins, Angew. Chem. Int. Ed. 2021, 60, 1959–1966.

17. Q. Zheng*, H. Xu*, H. Wang, W.H. Du, N. Wang, H. Xiong, Y. Gu, L. Noodleman, K.B. Sharpless#, G. Yang#, P. Wu#, Sulfur [18F]Fluoride Exchange Click Chemistry Enabled Ultrafast Late-Stage Radiosynthesis, J. Am. Chem. Soc. 2021, 143, 3753–3763.

18. H. Xu*, Y. Gu*, S. Zhang, H. Xiong, F. Ma, F. Lu, Q. Ji, L. Liu, P. Ma, W. Hou#, G. Yang#, R.A. Lerner#, A Chemistry for Incorporation of Selenium into DNAEncoded Libraries, Angew. Chem. Int. Ed. 2020, 59, 13273–13280.

19. H. Xu*, F. Ma*, N. Wang, W. Hou, H. Xiong, F. Lu, J. Li, S. Wang, P. Ma, G. Yang#, R.A. Lerner#, DNAEncoded Libraries: Aryl Fluorosulfonates as Versatile Electrophiles Enabling Facile OnDNA Suzuki, Sonogashira, and Buchwald Reactions, Adv. Sci. 2019, 6, 1901551.

20. P. Ma*, H. Xu*, J. Li*, F. Lu, F. Ma, S. Wang, H. Xiong, W. Wang, D. Buratto, F. Zonta, N. Wang, K. Liu, T. Hua, Z. Liu, G. Yang#, R.A. Lerner#, Functionality independent DNA encoding of complex natural products, Angew. Chem. Int. Ed. 2019, 58, 9254-9261.